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Found 27 of affinity data for UniProtKB/TrEMBL: O02824
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)
Affinity DataKi:  275nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM66983(6-chloranyl-3-methyl-1,2,4,5-tetrahydro-3-benzazep...)
Affinity DataKi:  900nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50026636(17alpha-hydroxy-20alpha-yohimban-16beta-carboxylic...)
Affinity DataKi:  1.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50026636(17alpha-hydroxy-20alpha-yohimban-16beta-carboxylic...)
Affinity DataKi:  1.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50019848(2-(2,3-dihydro-1,4-benzodioxin-2-yl)-4,5-dihydro-1...)
Affinity DataKi:  2.30E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50026636(17alpha-hydroxy-20alpha-yohimban-16beta-carboxylic...)
Affinity DataKi:  4.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82472(BW-723C86 | CAS_5311036 | NSC_5311036)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82472(BW-723C86 | CAS_5311036 | NSC_5311036)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50474666(CHEMBL321644)
Affinity DataEC50:  2.82E+3nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50474633(CHEMBL111496)
Affinity DataEC50:  631nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50118702(2-Amino-1-(2,5-dimethoxy-phenyl)-ethanol | CHEMBL1...)
Affinity DataEC50:  7.08E+3nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50022722((+)2-Amino-1-phenyl-propan-1-ol | (1R, 2R)-2-Amino...)
Affinity DataEC50:  2.34E+5nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50474634(CHEMBL322492)
Affinity DataEC50:  1.91E+4nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50474652(CHEMBL325897)
Affinity DataEC50:  5.62E+3nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50118703(CHEMBL109783 | N-[5-(4,5-Dihydro-1H-imidazol-2-yl)...)
Affinity DataEC50:  9.30nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50474654(CHEMBL323402)
Affinity DataEC50:  275nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50474650(CHEMBL111537)
Affinity DataEC50:  6.76E+3nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50474648(CHEMBL109848)
Affinity DataEC50:  1.29E+3nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50474660(CHEMBL111771)
Affinity DataEC50:  66nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50474670(CHEMBL111584)
Affinity DataEC50:  5.50E+3nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataEC50:  603nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50487266(CHEMBL2261355)
Affinity DataEC50:  170nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50474671(CHEMBL111554)
Affinity DataEC50:  447nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50474643(CHEMBL111734)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at rabbit urethra adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(RABBIT)
Smith Kline & French Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50474630(CHEMBL108804)
Affinity DataEC50:  17nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article